Publication Details (including relevant citation information):
D.Giribone, C. Felicini, E.Fontana
Synthesis and Applications of Isotopically Labelled Compounds, Volume 7 (2000) 236-239, John Wiley & Sons LTD
In this paper we describe the case of three substituted pyrazines for which the original laboratory-scale synthesis was completely reviewed and modified. The preparation of the radiolabelled analogues in a cost-efficient manner starting from a common intermediate by means of the Mitsunobu reaction as the key step performed with a parallel synthesis equipment. The labelling approach is also discussed.
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