Danilo Giribone - Synthesis of PNU-243922 Labelled with carbon-14

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  Publication Details (including relevant citation   information):

  C. Felicini,   E.Fontana, D.Giribone, B.M.Nilsson, K.O Osterlund, and   A.Paptchikhine

  Journal of   Labelled Compounds and   Radiopharmaceuticals, 46 (2003) 85-92


  The arylpiperazine PNU-243922 (1) has been   labelled with 14C. A two-step sequence starting from   the 14C labelled alcohol 6a led to   radiochemically pure (>98%) [14C]PNU-243922 with a   specific activity of 546 MBq/mmol

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